Pseudomonas aeruginosa FabF C164A mutant in complex with(S)-2-(1H-pyrazole-3-carboxamido)butanoic acid
收藏Protein Data Bank Japan2025-05-07 更新2026-04-19 收录
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Pseudomonas aeruginosa FabF C164A mutant in complex with(S)-2-(1H-pyrazole-3-carboxamido)butanoic acid Descriptor: (2~{S})-2-(1~{H}-pyrazol-3-ylcarbonylamino)butanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 2, CHLORIDE ION, ... Authors: Georgiou, C, Brenk, R, Yadrykhinsky, V, Espeland, L.O. Deposit date: 2023-06-17 Release date: 2024-01-10 Last modified: 2025-05-07 Method: X-RAY DIFFRACTION (1.78 Å) Cite: Towards new antibiotics: P. aeruginosa FabF ligands discovered by crystallographic fragment screening followed by hit expansion. Eur.J.Med.Chem., 291, 2025
创建时间:
2023-06-17



