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Pseudomonas aeruginosa FabF C164A mutant in complex with N-isopropyl-1H-imidazole-4-carboxamide

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Protein Data Bank Japan2025-05-07 更新2026-04-25 收录
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https://pdbj.org/mine/summary/8pd1
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Pseudomonas aeruginosa FabF C164A mutant in complex with N-isopropyl-1H-imidazole-4-carboxamide Descriptor: 3-oxoacyl-[acyl-carrier-protein] synthase 2, CHLORIDE ION, DIMETHYL SULFOXIDE, ... Authors: Georgiou, C, Brenk, R, Yadrykhinsky, V, Espeland, L.O. Deposit date: 2023-06-11 Release date: 2024-01-10 Last modified: 2025-05-07 Method: X-RAY DIFFRACTION (1.87 Å) Cite: Towards new antibiotics: P. aeruginosa FabF ligands discovered by crystallographic fragment screening followed by hit expansion. Eur.J.Med.Chem., 291, 2025
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2023-06-11
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