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Crystal Structure of human glutaminase with macrocyclic inhibitor

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6lox
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资源简介:
Crystal Structure of human glutaminase with macrocyclic inhibitor Descriptor: (E)-15,22-Dioxa-4,11-diaza-5(2,5)-thiadiazola-10(3,6)-pyridazina-1,14(1,3)-dibenzenacyclodocosaphan-18-ene-3,12-dione, Glutaminase kidney isoform, mitochondrial Authors: Bian, J, Li, Z, Xu, X, Wang, J, Li, L. Deposit date: 2020-01-07 Release date: 2021-01-13 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (3.2 Å) Cite: Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site. J.Med.Chem., 64, 2021
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2020-01-07
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