17beta-hydroxysteroid dehydrogenase 14 variant T205 in complex with a non-steroidal quinoline based inhibitor
收藏Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5o72
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17beta-hydroxysteroid dehydrogenase 14 variant T205 in complex with a non-steroidal quinoline based inhibitor Descriptor: 17-beta-hydroxysteroid dehydrogenase 14, 2-azanyl-~{N}-[2-(4-fluoranyl-3-oxidanyl-phenyl)carbonylquinolin-7-yl]ethanamide, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... Authors: Bertoletti, N, Braun, F, Heine, A, Klebe, G, Marchais-Oberwinkler, S. Deposit date: 2017-06-07 Release date: 2018-06-06 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (1.91 Å) Cite: Structure-based design and profiling of novel 17 beta-HSD14 inhibitors. Eur J Med Chem, 155, 2018
创建时间:
2017-06-07



