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CRYSTAL STRUCTURE OF HUMAN PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH FARNESYL DIPHOSPHATE AND THE PEPTIDOMIMETIC INHIBITOR L-739,750

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Protein Data Bank Japan2023-08-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1jcq
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CRYSTAL STRUCTURE OF HUMAN PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH FARNESYL DIPHOSPHATE AND THE PEPTIDOMIMETIC INHIBITOR L-739,750 Descriptor: 2(S)-{2(S)-[2(R)-AMINO-3-MERCAPTO]PROPYLAMINO-3(S)-METHYL}PENTYLOXY-3-PHENYLPROPIONYLMETHIONINE SULFONE, ACETIC ACID, FARNESYL DIPHOSPHATE, ... Authors: Long, S.B, Casey, P.J, Beese, L.S. Deposit date: 2001-06-11 Release date: 2001-11-02 Last modified: 2023-08-16 Method: X-RAY DIFFRACTION (2.3 Å) Cite: The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98, 2001
创建时间:
2001-06-11
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