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Synthesis and biological evaluation of new triazolo and imidazolopyridine RORgt inverse agonists

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Synthesis and biological evaluation of new triazolo and imidazolopyridine RORgt inverse agonists Descriptor: Nuclear receptor ROR-gamma, ~{N}-[8-[[(3~{S})-4-cyclopentylcarbonyl-3-methyl-piperazin-1-yl]methyl]-7-methyl-imidazo[1,2-a]pyridin-6-yl]-2-methyl-pyrimidine-5-carboxamide Authors: Kallen, J. Deposit date: 2016-10-31 Release date: 2016-12-14 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.77 Å) Cite: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine ROR gamma t Inverse Agonists. ChemMedChem, 11, 2016
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2016-10-31
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