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Aurora A kinase bound to a highly selective imidazopyridine inhibitor

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4byi
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资源简介:
Aurora A kinase bound to a highly selective imidazopyridine inhibitor Descriptor: (S)-N-((1-(6-chloro-2-(1,3-dimethyl-1H-pyrazol-4-yl)-3H-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamide, AURORA KINASE A Authors: Joshi, A, Kosmopoulou, M, Bayliss, R. Deposit date: 2013-07-19 Release date: 2013-11-20 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Aurora Isoform Selectivity: Design and Synthesis of Imidazo[4,5-B]Pyridine Derivatives as Highly Selective Inhibitors of Aurora-A Kinase in Cells. J.Med.Chem., 56, 2013
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2013-07-19
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