five

mGluR2 ECD and mGluR3 ECD complex with ligands

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Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
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mGluR2 ECD and mGluR3 ECD complex with ligands Descriptor: (1S,2S,5R,6S)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid, IODIDE ION, Metabotropic glutamate receptor 3 Authors: Clawson, D.K. Deposit date: 2014-12-15 Release date: 2015-02-11 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (2.26 Å) Cite: Synthesis and Pharmacological Characterization of C4-Disubstituted Analogs of 1S,2S,5R,6S-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate: Identification of a Potent, Selective Metabotropic Glutamate Receptor Agonist and Determination of Agonist-Bound Human mGlu2 and mGlu3 Amino Terminal Domain Structures. J.Med.Chem., 58, 2015
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2014-12-15
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