five

InhA in complex with a DNA encoded library hit

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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InhA in complex with a DNA encoded library hit Descriptor: (2S,4S)-N-methyl-4-[[(2S,3R)-3-[(2-methylpropan-2-yl)oxy]-2-[[4-(pyrazol-1-ylmethyl)phenyl]carbonylamino]butanoyl]amino]-1-(phenylcarbonyl)pyrrolidine-2-carboxamide, ENOYL-ACYL CARRIER PROTEIN REDUCTASE, MAGNESIUM ION, ... Authors: Read, J.A, Breed, J. Deposit date: 2016-03-22 Release date: 2016-11-30 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.79 Å) Cite: Discovery of Cofactor-Specific, Bactericidal Mycobacterium Tuberculosis Inha Inhibitors Using DNA-Encoded Library Technology Proc.Natl.Acad.Sci.USA, 113, 2016
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2016-03-22
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