TTK kinase domain in complex with MPI-0479605
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5n7v
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TTK kinase domain in complex with MPI-0479605 Descriptor: 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, Dual specificity protein kinase TTK, ~{N}6-cyclohexyl-~{N}2-(2-methyl-4-morpholin-4-yl-phenyl)-7~{H}-purine-2,6-diamine Authors: Uitdehaag, J, Willemsen-Seegers, N, Zaman, G.J.R. Deposit date: 2017-02-21 Release date: 2017-05-31 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.52 Å) Cite: Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity. J. Mol. Biol., 429, 2017
创建时间:
2017-02-21



