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tRNA Guanine Transglycosylase in complex with disubstituted lin-benzoguanine inhibitor

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Protein Data Bank Japan2025-11-12 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4gkt
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tRNA Guanine Transglycosylase in complex with disubstituted lin-benzoguanine inhibitor Descriptor: 6-amino-4-{2-[(cyclopentylmethyl)amino]ethyl}-2-[(2-phenylethyl)amino]-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one, GLYCEROL, Queuine tRNA-ribosyltransferase, ... Authors: Immekus, F, Klebe, G. Deposit date: 2012-08-13 Release date: 2013-09-04 Last modified: 2025-11-12 Method: X-RAY DIFFRACTION (1.53 Å) Cite: High-affinity inhibitors of Zymomonas mobilis tRNA-guanine transglycosylase through convergent optimization. Acta Crystallogr.,Sect.D, 69, 2013
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2012-08-13
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