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Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor Descriptor: 1-[[4-fluoranyl-3-[4-[2,2,2-tris(fluoranyl)ethyl]piperazin-1-yl]carbonyl-phenyl]methyl]quinazoline-2,4-dione, Poly [ADP-ribose] polymerase 1 Authors: Cao, R, Wang, Y.L, Zhou, J, Huang, N, Xu, B.L. Deposit date: 2016-12-11 Release date: 2017-01-25 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor To Be Published
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2016-12-11
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