Crystal structure of BRD2(BD2) W370F mutant with ligand I-BET 762 bound
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Crystal structure of BRD2(BD2) W370F mutant with ligand I-BET 762 bound Descriptor: 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide, Bromodomain-containing protein 2, GLYCEROL, ... Authors: Tallant, C, Baud, M, Lin-Shiao, E, Chirgadze, D.Y, Ciulli, A. Deposit date: 2015-08-26 Release date: 2015-11-11 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.5 Å) Cite: New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition. J.Med.Chem., 59, 2016
创建时间：
2015-08-26
