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Tankyrase-2 in complex with compound 40c

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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Tankyrase-2 in complex with compound 40c Descriptor: 2-[4,6-difluoro-1-(2-hydroxyethyl)-1,2-dihydro-1'H-spiro[indole-3,4'-piperidin]-1'-yl]-5,6,7,8-tetrahydroquinazolin-4(3H)-one, GLYCEROL, PHOSPHATE ION, ... Authors: Niwa, H, Shirai, F, Sato, S, Yoshimoto, N, Tsumura, T, Okue, M, Shirouzu, M, Seimiya, H, Umehara, T. Deposit date: 2018-04-19 Release date: 2019-04-03 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. J. Med. Chem., 62, 2019
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2018-04-19
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