PLK1 SURFACE ENTROPY REDUCTION (SER) MUTANT IN COMPLEX WITH INHIBITOR BI 2536
收藏Protein Data Bank Japan2025-12-10 更新2026-04-19 收录
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PLK1 SURFACE ENTROPY REDUCTION (SER) MUTANT IN COMPLEX WITH INHIBITOR BI 2536 Descriptor: 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, GLYCEROL, SULFATE ION, ... Authors: Hillig, R.C, Schulze, V.K, Siemeister, G, Schmitz, A.A, Eberspaecher, U. Deposit date: 2025-04-28 Release date: 2025-11-26 Last modified: 2025-12-10 Method: X-RAY DIFFRACTION (2.84 Å) Cite: Polo-like kinase 1-inhibitor co-complex structures via the surface-entropy reduction approach and a DARPin-assisted approach. Acta Crystallogr D Struct Biol, 81, 2025
创建时间:
2025-04-28



