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Human peroxisome proliferator-activated receptor (PPAR) delta ligand binding domain in complex with a synthetic partial agonist JK122

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Protein Data Bank Japan2023-11-29 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7vwe
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Human peroxisome proliferator-activated receptor (PPAR) delta ligand binding domain in complex with a synthetic partial agonist JK122 Descriptor: 5-[4-butoxy-3-[[[2-fluoranyl-4-(trifluoromethyl)phenyl]carbonylamino]methyl]phenyl]-4,6-dimethyl-pyridine-3-carboxylic acid, Peroxisome proliferator-activated receptor delta, heptyl beta-D-glucopyranoside Authors: Oyama, T, Miyachi, H. Deposit date: 2021-11-10 Release date: 2022-02-09 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (3 Å) Cite: Crystal structures of the ligand-binding domain of human peroxisome proliferator-activated receptor delta in complexes with phenylpropanoic acid derivatives and a pyridine carboxylic acid derivative. Acta Crystallogr.,Sect.F, 78, 2022
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2021-11-10
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