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DYRK1A in complex with XMD14-124

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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DYRK1A in complex with XMD14-124 Descriptor: Dual specificity tyrosine-phosphorylation-regulated kinase 1A, [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone Authors: Rothweiler, U. Deposit date: 2017-09-19 Release date: 2018-08-29 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Novel Scaffolds for Dual Specificity Tyrosine-Phosphorylation-Regulated Kinase (DYRK1A) Inhibitors. J. Med. Chem., 61, 2018
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2017-09-19
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