Human Tankyrase 2 - Catalytic PARP domain in complex with an inhibitor
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Human Tankyrase 2 - Catalytic PARP domain in complex with an inhibitor Descriptor: 2-[4-(4-fluorophenyl)piperazin-1-yl]-6-methylpyrimidin-4(3H)-one, SULFATE ION, Tankyrase-2, ... Authors: Karlberg, T, Siponen, M.I, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Kotenyova, T, Kouznetsova, E, Moche, M, Nordlund, P, Nyman, T, Persson, C, Schutz, P, Sehic, A, Thorsell, A.G, Tresaugues, L, Van Den Berg, S, Wahlberg, E, Weigelt, J, Welin, M, Schuler, H, Structural Genomics Consortium (SGC) Deposit date: 2010-09-29 Release date: 2010-10-20 Last modified: 2023-11-01 Method: X-RAY DIFFRACTION (2.49 Å) Cite: Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors Nat.Biotechnol., 30, 2012
创建时间:
2010-09-29



