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MBX2319 bound structure of bacterial efflux pump.

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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MBX2319 bound structure of bacterial efflux pump. Descriptor: 3,3-dimethyl-8-morpholin-4-yl-6-(2-phenylethylsulfanyl)-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile, DARPin, Multidrug efflux pump subunit AcrB,Multidrug efflux pump subunit AcrB Authors: Sjuts, H, Ornik, A.R, Pos, K.M. Deposit date: 2015-11-09 Release date: 2016-04-06 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives. Proc.Natl.Acad.Sci.USA, 113, 2016

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2015-11-09
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