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RSK2 T493M C-Terminal Kinase Domain in Complex with RMM58

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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RSK2 T493M C-Terminal Kinase Domain in Complex with RMM58 Descriptor: (2Z)-2-(1H-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1H-indazol-5-yl]prop-2-enenitrile, Ribosomal protein S6 kinase alpha-3, SODIUM ION Authors: Miller, R.M, Taunton, J. Deposit date: 2013-08-16 Release date: 2014-10-22 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Design of reversible, cysteine-targeted Michael acceptors guided by kinetic and computational analysis. J.Am.Chem.Soc., 136, 2014

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2013-08-16
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