Crystal structure of PPAR gamma ligand binding domain in complex with a novel partial agonist GQ-16
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Crystal structure of PPAR gamma ligand binding domain in complex with a novel partial agonist GQ-16 Descriptor: (5Z)-5-(5-bromo-2-methoxybenzylidene)-3-(4-methylbenzyl)-1,3-thiazolidine-2,4-dione, Nuclear receptor coactivator 1, Peroxisome proliferator-activated receptor gamma Authors: Rajagopalan, S, Webb, P, Baxter, J.D, Brennan, R.G, Phillips, K.J. Deposit date: 2011-07-19 Release date: 2012-05-23 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2.1 Å) Cite: GQ-16, a novel peroxisome proliferator-activated receptor (PPAR gamma) ligand, promotes insulin sensitization without weight gain. J.Biol.Chem., 287, 2012
创建时间:
2011-07-19



