Leishmania major N-myristoyltransferase in complex with thienopyrimidine inhibitor IMP-0000096
收藏Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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Leishmania major N-myristoyltransferase in complex with thienopyrimidine inhibitor IMP-0000096 Descriptor: 3-[[6-tert-butyl-2-[methyl-[(3S)-1-methylpyrrolidin-3-yl]amino]thieno[3,2-d]pyrimidin-4-yl]-methyl-amino]propanenitrile, Glycylpeptide N-tetradecanoyltransferase, MAGNESIUM ION, ... Authors: Brannigan, J.A. Deposit date: 2019-01-01 Release date: 2020-05-06 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.49 Å) Cite: Novel Thienopyrimidine Inhibitors of Leishmania N -Myristoyltransferase with On-Target Activity in Intracellular Amastigotes. J.Med.Chem., 63, 2020
创建时间:
2019-01-01



