five

HSP90 WITH indazole derivative

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5lo0
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资源简介:
HSP90 WITH indazole derivative Descriptor: Heat shock protein HSP 90-alpha, [2-azanyl-6-[4,5-bis(fluoranyl)-2-(4-methylpiperazin-1-yl)sulfonyl-phenyl]quinazolin-4-yl]-(1,3-dihydroisoindol-2-yl)methanone Authors: Graedler, U, Amaral, M, Schuetz, D. Deposit date: 2016-08-08 Release date: 2017-11-29 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Ligand Desolvation Steers On-Rate and Impacts Drug Residence Time of Heat Shock Protein 90 (Hsp90) Inhibitors. J. Med. Chem., 61, 2018
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2016-08-08
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