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IRAK4 in complex with inhibitor

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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IRAK4 in complex with inhibitor Descriptor: Interleukin-1 receptor-associated kinase 4, N-[(2R)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide, SULFATE ION Authors: Ghosh, K, Bose, S. Deposit date: 2020-02-12 Release date: 2020-11-25 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.19 Å) Cite: Optimization of Nicotinamides as Potent and Selective IRAK4 Inhibitors with Efficacy in a Murine Model of Psoriasis. Acs Med.Chem.Lett., 11, 2020

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2020-02-12
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