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Crystal structure of HsaD bound to 3,5-dichloro-4-hydroxybenzenesulphonic acid

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal structure of HsaD bound to 3,5-dichloro-4-hydroxybenzenesulphonic acid Descriptor: 3,5-dichloro-4-hydroxybenzene-1-sulfonic acid, 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase Authors: Ryan, A, Polycarpou, E, Lack, N.A, Evangelopoulos, D, Sieg, C, Halman, A, Bhakta, S, Sinclair, A, Eleftheriadou, O, McHugh, T.D, Keany, S, Lowe, E, Ballet, R, Abihammad, A, Ciulli, A, Sim, E. Deposit date: 2016-05-16 Release date: 2017-04-05 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.68 Å) Cite: Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. Br. J. Pharmacol., 174, 2017

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2016-05-16
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