遇见数据集

Toxoplasma Gondii CDPK1 in complex with inhibitor GXJ-237

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Protein Data Bank Japan2026-05-20 更新2026-03-21 收录
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Toxoplasma Gondii CDPK1 in complex with inhibitor GXJ-237 Descriptor: 3-(3-chlorophenoxy)-1-[(piperidin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine, CALCIUM ION, Calmodulin-domain protein kinase 1 Authors: El Bakkouri, M, Lovato, D, Loppnau, P, Lin, Y.H, Rutaganaria, F, Lopez, M.S, Shokat, L, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Sibley, D, Walker, J.R, Structural Genomics Consortium (SGC) Deposit date: 2017-06-21 Release date: 2017-07-19 Last modified: 2026-05-20 Method: X-RAY DIFFRACTION (2 Å) Cite: Inhibition of Calcium Dependent Protein Kinase 1 (CDPK1) by Pyrazolopyrimidine Analogs Decreases Establishment and Reoccurrence of Central Nervous System Disease by Toxoplasma gondii. J.Med.Chem., 60, 2017

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2017-06-21
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