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Crystal Structure of JAK2 complexed with a potent quinoxaline ATP site inhibitor

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Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
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资源简介:
Crystal Structure of JAK2 complexed with a potent quinoxaline ATP site inhibitor Descriptor: 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1H-pyrazol-4-yl)quinoxaline, Tyrosine-protein kinase JAK2 Authors: Tavares, G.A, Gerspacher, M, Kroemer, M, Scheufler, C. Deposit date: 2009-11-19 Release date: 2010-07-21 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Potent and Selective Inhibition of Polycythemia by the Quinoxaline JAK2 Inhibitor NVP-BSK805 Mol.Cancer Ther., 9, 2010
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2009-11-19
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