Pi3K alpha lipid kinase with Active Site Inhibitor
收藏Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4ykn
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Pi3K alpha lipid kinase with Active Site Inhibitor Descriptor: 3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acid, Phosphatidylinositol 3-kinase regulatory subunit alpha,Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform fusion protein Authors: Elkins, P.A. Deposit date: 2015-03-04 Release date: 2015-06-17 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Discovery of a Potent Class of PI3K alpha Inhibitors with Unique Binding Mode via Encoded Library Technology (ELT). Acs Med.Chem.Lett., 6, 2015
创建时间:
2015-03-04



