Crystal structure of human tankyrase 2 in complex with EB-47
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Crystal structure of human tankyrase 2 in complex with EB-47 Descriptor: 2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide, GLYCEROL, SULFATE ION, ... Authors: Haikarainen, T, Narwal, M, Lehtio, L. Deposit date: 2013-04-17 Release date: 2013-12-11 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Evaluation and Structural Basis for the Inhibition of Tankyrases by Parp Inhibitors Acs Med.Chem.Lett., 5, 2014
创建时间:
2013-04-17



