five

MPS1 kinase with 3-aminopyridin-2-one inhibitors

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4cv8
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MPS1 kinase with 3-aminopyridin-2-one inhibitors Descriptor: 1,2-ETHANEDIOL, 3-amino-5-(1-methyl-1H-pyrazol-4-yl)pyridin-2(1H)-one, DUAL SPECIFICITY PROTEIN KINASE TTK Authors: Fearon, D, Bavetsias, V, Bayliss, R, Schmitt, J, Westwood, I.M, vanMontfort, R.L.M, Jones, K. Deposit date: 2014-03-24 Release date: 2015-04-08 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (3 Å) Cite: Protein Kinase Selectivity of a 3-Aminopyridin-2- One Based Fragment Library, Identification of 3-Amino-5-(Pyridin-4-Yl)Pyridin-2(1H)-One as a Novel Scaffold for Mps1 Inhibition To be Published
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2014-03-24
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