Plasmodium vivax N-myristoyltransferase in complex with a pyrazole sulphonamide inhibitor.
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Plasmodium vivax N-myristoyltransferase in complex with a pyrazole sulphonamide inhibitor. Descriptor: 2,6-dichloro-4-(2-piperazin-1-ylpyridin-4-yl)-N-(1,3,5-trimethyl-1H-pyrazol-4-yl)benzenesulfonamide, 2-oxopentadecyl-CoA, CHLORIDE ION, ... Authors: Wright, M.H, Clough, B, Rackham, M.D, Brannigan, J.A, Grainger, M, Bottrill, A.R, Heal, W.P, Broncel, M, Serwa, R.A, Mann, D, Leatherbarrow, R.J, Wilkinson, A.J, Holder, A.A, Tate, E.W. Deposit date: 2012-10-13 Release date: 2014-01-15 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.89 Å) Cite: Validation of N-Myristoyltransferase as an Antimalarial Drug Target Using an Integrated Chemical Biology Approach. Nat.Chem., 6, 2014
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2012-10-13



