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M. thermoresistible GuaB2 delta-CBS in complex with inhibitor Compound 18 (VCC399134)

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Protein Data Bank Japan2026-04-15 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6d4r
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M. thermoresistible GuaB2 delta-CBS in complex with inhibitor Compound 18 (VCC399134) Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase,Inosine-5'-monophosphate dehydrogenase, [4-(isoquinoline-5-sulfonyl)piperazin-1-yl](3-nitrophenyl)methanone Authors: Ascher, D.B, Pacitto, A, Blundell, T.L. Deposit date: 2018-04-18 Release date: 2019-05-01 Last modified: 2026-04-15 Method: X-RAY DIFFRACTION (1.34 Å) Cite: Synthesis and Structure-Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH. Eur.J.Med.Chem., 174, 2019
创建时间:
2018-04-18
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