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Crystal structure of human ATAD2 bromodomain in complex with 3-methyl- 8-piperidin-4-ylamino-1,2-dihydro-1,7-naphthyridin-2-one hydrochloride

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of human ATAD2 bromodomain in complex with 3-methyl- 8-piperidin-4-ylamino-1,2-dihydro-1,7-naphthyridin-2-one hydrochloride Descriptor: 1,2-ETHANEDIOL, 3-methyl-8-[(piperidin-4-yl)amino]-1,2-dihydro-1,7-naphthyridin-2-one, ATPASE FAMILY AAA DOMAIN-CONTAINING PROTEIN 2, ... Authors: Chung, C, Bamborough, P, Demont, E. Deposit date: 2015-06-20 Release date: 2015-07-22 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.97 Å) Cite: Fragment-Based Discovery of Low-Micromolar Atad2 Bromodomain Inhibitors. J.Med.Chem., 58, 2015
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2015-06-20
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