CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 17528462
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https://pdbj.org/mine/summary/5ti7
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CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 17528462 Descriptor: 1,2-ETHANEDIOL, 5-bromo-2-methoxy-N-(3-(2-oxopyrrolidin-1-yl)phenyl)benzenesulfonamide, Bromodomain-containing protein 4 Authors: Zhu, J.-Y, Ember, S.W.J, Schonbrunn, E. Deposit date: 2016-10-01 Release date: 2017-08-09 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations. ACS Omega, 2, 2017
创建时间:
2016-10-01



