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Crystal structure of MEK1 in complex with fragment 18

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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资源简介:
Crystal structure of MEK1 in complex with fragment 18 Descriptor: 7-choro-6-[(3R)-pyrrolidin-3-ylmethoxy]isoquinolin-1(2H)-one, DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1 Authors: Amaning, K, Lowinsky, M, Vallee, F, Steier, V, Marcireau, C, Ugolini, A, Delorme, C, McCort, G, Andouche, C, Vougier, S, Llopart, S, Halland, N, Rak, A. Deposit date: 2013-02-04 Release date: 2013-05-22 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.2 Å) Cite: The Use of Virtual Screening and Differential Scanning Fluorimetry for the Rapid Identification of Fragments Active Against Mek1. Bioorg.Med.Chem.Lett., 23, 2013
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2013-02-04
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