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Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with dasatinib

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with dasatinib Descriptor: 1,2-ETHANEDIOL, Ephrin type-A receptor 2, N-(2-CHLORO-6-METHYLPHENYL)-2-({6-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]-2-METHYLPYRIMIDIN-4-YL}AMINO)-1,3-THIAZOLE-5-CARBOXAMIDE Authors: Kudlinzki, D, Linhard, V.L, Gande, S.L, Sreeramulu, S, Saxena, K, Heinzlmeir, S, Medard, G, Kuester, B, Schwalbe, H. Deposit date: 2016-02-21 Release date: 2016-11-09 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.228 Å) Cite: Chemical Proteomics and Structural Biology Define EPHA2 Inhibition by Clinical Kinase Drugs. ACS Chem. Biol., 11, 2016
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2016-02-21
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