遇见数据集

KAT6A IN COMPLEX WITH SMALL MOLECULE INHIBITOR BAY-184

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Protein Data Bank Japan2024-11-27 更新2026-04-19 收录
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KAT6A IN COMPLEX WITH SMALL MOLECULE INHIBITOR BAY-184 Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 6-(dimethylamino)-~{N}-(2-phenylphenyl)sulfonyl-1-benzofuran-2-carboxamide, Histone acetyltransferase KAT6A, ... Authors: Hillig, R.C, Puetter, V. Deposit date: 2024-06-04 Release date: 2024-11-06 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (2.69 Å) Cite: Discovery and Characterization of BAY-184: A New Potent and Selective Acylsulfonamide-Benzofuran In Vivo -Active KAT6AB Inhibitor. J.Med.Chem., 67, 2024

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2024-06-04
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