EthR2 in complex with compound 1 (BDM14272)
收藏Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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EthR2 in complex with compound 1 (BDM14272) Descriptor: (1~{S},5~{R})-8-[2-(4-chlorophenyl)ethyl]-8-azabicyclo[3.2.1]octan-3-one, Probable transcriptional regulatory protein Authors: Wintjens, R, Wohlkonig, A, Tanina, A. Deposit date: 2018-09-28 Release date: 2019-02-27 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.45 Å) Cite: A fragment-based approach towards the discovery of N-substituted tropinones as inhibitors of Mycobacterium tuberculosis transcriptional regulator EthR2. Eur J Med Chem, 167, 2019
创建时间:
2018-09-28



