3.06A COMPLEX OF S.AUREUS GYRASE with imidazopyrazinone T1 AND DNA
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3.06A COMPLEX OF S.AUREUS GYRASE with imidazopyrazinone T1 AND DNA Descriptor: 7-[(3~{S})-3-azanylpyrrolidin-1-yl]-5-cyclopropyl-8-fluoranyl-imidazo[1,2-a]quinoxalin-4-one, DNA (5'-D(*GP*AP*GP*AP*GP*TP*AP*T*GP*GP*CP*CP*AP*TP*AP*CP*TP*CP*T)-3'), DNA gyrase subunit A, ... Authors: Bax, B.D, Germe, T, Basque, E, Maxwell, A. Deposit date: 2018-02-14 Release date: 2018-04-04 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (3.06 Å) Cite: A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance. Nucleic Acids Res., 46, 2018
创建时间:
2018-02-14



