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Hsp90 Alpha N-terminal Domain in Complex with an Inhibitor 6-Hydroxy-3-(3-methyl-benzyl)-1H-indazole-5-carboxylic acid benzyl-methyl-amide

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Protein Data Bank Japan2024-03-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4efu
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资源简介:
Hsp90 Alpha N-terminal Domain in Complex with an Inhibitor 6-Hydroxy-3-(3-methyl-benzyl)-1H-indazole-5-carboxylic acid benzyl-methyl-amide Descriptor: Heat shock protein HSP 90-alpha, N-benzyl-6-hydroxy-N-methyl-3-(3-methylbenzyl)-1H-indazole-5-carboxamide, SULFATE ION Authors: Musil, D, Lehmann, M, Graedler, U, Buchstaller, H.-P. Deposit date: 2012-03-30 Release date: 2012-06-27 Last modified: 2024-03-20 Method: X-RAY DIFFRACTION (2 Å) Cite: Fragment-based discovery of hydroxy-indazole-carboxamides as novel small molecule inhibitors of Hsp90 Bioorg.Med.Chem.Lett., 22, 2012
创建时间:
2012-03-30
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