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Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with Compound 2i

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with Compound 2i Descriptor: 1,2-ETHANEDIOL, 2-[(3~{R})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acid, Ephrin type-A receptor 2 Authors: Kudlinzki, D, Linhard, V.L, Witt, K, Gande, S.L, Saxena, K, Heinzlmeir, S, Medard, G, Kuester, B, Schwalbe, H. Deposit date: 2017-03-31 Release date: 2017-06-07 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.408 Å) Cite: Chemoproteomics-Aided Medicinal Chemistry for the Discovery of EPHA2 Inhibitors. ChemMedChem, 12, 2017
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2017-03-31
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