Crystal structure of drug resistant SRC kinase domain with irreversible inhibitor
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Crystal structure of drug resistant SRC kinase domain with irreversible inhibitor Descriptor: (2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide, Proto-oncogene tyrosine-protein kinase Src Authors: Michalczyk, A, Rode, H.B, Gruetter, C, Rauh, D. Deposit date: 2007-07-26 Release date: 2008-03-11 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.38 Å) Cite: Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR. Bioorg.Med.Chem., 16, 2008
创建时间:
2007-07-26



