five

Crystal structure of autotaxin in complex with BI-2545

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Crystal structure of autotaxin in complex with BI-2545 Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3,6,9,12,15-PENTAOXAHEPTADECANE, CALCIUM ION, ... Authors: Hoerer, S. Deposit date: 2017-07-17 Release date: 2018-01-03 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.66 Å) Cite: Discovery of BI-2545: A Novel Autotaxin Inhibitor That Significantly Reduces LPA Levels in Vivo. ACS Med Chem Lett, 8, 2017
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2017-07-17
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