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HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 28

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Protein Data Bank Japan2024-04-03 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7lq1
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HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 28 Descriptor: CHLORIDE ION, N-(5-(6-(2-((2S,6R)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamide, Phosphatidylinositol 3-kinase regulatory subunit alpha, ... Authors: Lesburg, C.A, Augustin, M. Deposit date: 2021-02-12 Release date: 2022-02-16 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.96 Å) Cite: Discovery of a new series of PI3K-delta inhibitors from Virtual Screening. Bioorg.Med.Chem.Lett., 42, 2021
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2021-02-12
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