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Fragment-Based Design of novel Estrogen Receptor Ligands

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Fragment-Based Design of novel Estrogen Receptor Ligands Descriptor: 2-(trifluoroacetyl)-1,2,3,4-tetrahydroisoquinolin-6-ol, Estrogen receptor beta, Nuclear receptor coactivator 1 Authors: Moecklinghoff, S, van Otterlo, W.A, Rose, R, Fuchs, S, Dominguez Seoane, M, Waldmann, H, Ottmann, C, Brunsveld, L. Deposit date: 2010-08-27 Release date: 2011-03-16 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2.21 Å) Cite: Design and Evaluation of Fragment-Like Estrogen Receptor Tetrahydroisoquinoline Ligands from a Scaffold-Detection Approach. J.Med.Chem., 54, 2011
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2010-08-27
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