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Crystal Structure of Aurora-A L210C catalytic domain in complex with ASDO2

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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Crystal Structure of Aurora-A L210C catalytic domain in complex with ASDO2 Descriptor: (~{E})-~{N}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamide, Aurora kinase A, CHLORIDE ION, ... Authors: Bayliss, R, McIntyre, P.J. Deposit date: 2018-09-04 Release date: 2018-10-03 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Type II Kinase Inhibitors Targeting Cys-Gatekeeper Kinases Display Orthogonality with Wild Type and Ala/Gly-Gatekeeper Kinases. ACS Chem. Biol., 13, 2018
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2018-09-04
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