Protein kinase MKK7 in complex with 5-bromo-2-hydroxyphenyl-substituted pyrazolopyrimidine
收藏Protein Data Bank Japan2024-11-06 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7ovk
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Protein kinase MKK7 in complex with 5-bromo-2-hydroxyphenyl-substituted pyrazolopyrimidine Descriptor: 1-[(3~{R})-3-[4-azanyl-3-[1-(5-bromanyl-2-oxidanyl-phenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one, Dual specificity mitogen-activated protein kinase kinase 7, GLYCEROL Authors: Kleinboelting, S, Buehrmann, M, Mueller, M.P, Rauh, D. Deposit date: 2021-06-15 Release date: 2022-07-20 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Optimization of Covalent MKK7 Inhibitors via Crude Nanomole-Scale Libraries. J.Med.Chem., 65, 2022
创建时间:
2021-06-15



