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ANTI-TUMOR AGENT Y48 IN COMPLEX WITH TUBULIN

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Protein Data Bank Japan2026-03-04 更新2026-04-19 收录
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ANTI-TUMOR AGENT Y48 IN COMPLEX WITH TUBULIN Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-methyl-3-[(4-methylphenyl)sulfonylamino]-~{N}-[(6-methylpyridin-3-yl)methyl]benzamide, GUANOSINE-5'-DIPHOSPHATE, ... Authors: Du, T, Ji, M, Hou, Z, Lin, S, Zhang, J, Wu, D, Zhang, K, Lu, D, Xu, H, Chen, X. Deposit date: 2022-07-14 Release date: 2023-07-26 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Optimization of Benzamide Derivatives as Potent and Orally Active Tubulin Inhibitors Targeting the Colchicine Binding Site. J.Med.Chem., 65, 2022
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2022-07-14
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