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Crystal structure of PI3K-gamma in complex with pyrrolo-pyridine inhibitor 63

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Crystal structure of PI3K-gamma in complex with pyrrolo-pyridine inhibitor 63 Descriptor: 1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine], Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION Authors: Whittington, D.A, Tang, J, Yakowec, P. Deposit date: 2012-06-12 Release date: 2012-10-24 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (3 Å) Cite: Discovery and in Vivo Evaluation of Dual PI3K-beta/delta inhibitors J.Med.Chem., 55, 2012
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2012-06-12
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