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C-abl Kinase domain with the activator(cmpd29), N-(1-(3,4-dichlorophenyl)-4,5-dihydro-1H-pyrazol-3-yl)acetamide

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6npu
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C-abl Kinase domain with the activator(cmpd29), N-(1-(3,4-dichlorophenyl)-4,5-dihydro-1H-pyrazol-3-yl)acetamide Descriptor: 4-(4-METHYL-PIPERAZIN-1-YLMETHYL)-N-[4-METHYL-3-(4-PYRIDIN-3-YL-PYRIMIDIN-2-YLAMINO)-PHENYL]-BENZAMIDE, GLYCEROL, NONAETHYLENE GLYCOL, ... Authors: Campobasso, N. Deposit date: 2019-01-18 Release date: 2019-03-13 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.33 Å) Cite: Identification and Optimization of Novel Small c-Abl Kinase Activators Using Fragment and HTS Methodologies. J. Med. Chem., 62, 2019
创建时间:
2019-01-18
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